Bremazocine

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Bremazocine
Bremazocine.svg
Clinical data
Routes of
administration
Oral
ATC code
  • none
Identifiers
CAS Number
  • 75684-07-0
PubChem CID
  • 1223
IUPHAR/BPS
  • 1603
ChemSpider
  • 1186
UNII
  • ISF76M2DBE
ChEMBL
  • CHEMBL1165792 ☑Y
Chemical and physical data
Formula C20H29NO2
Molar mass 315.45 g/mol
3D model (JSmol)
  • Interactive image

Bremazocine is a κ-opioid receptor agonist related to pentazocine. It has potent and long-lasting analgesic and diuretic effects.[1] It has 200 times the activity of morphine, but appears to have no addictive properties and does not depress breathing.[2]

See also

References

  1. ^ Dortch-Carnes J, Potter DE (2005). "Bremazocine: a kappa-opioid agonist with potent analgesic and other pharmacologic properties". CNS Drug Reviews. 11 (2): 195–212. doi:10.1111/j.1527-3458.2005.tb00270.x. PMID 16007240.
  2. ^ Patrick, Graham (2013). An Introduction to Medicinal Chemistry (5th expanded ed.). Oxford University Press. p. 641. ISBN 0199697396.
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